Description

PT-141

Bremelanotide

Description

PT-141 is the isomer of Melanotan 2 without the C-end amide group, which

avoids characteristics such as sunburn stimulation and enhances

characteristics such as libido stimulation. Bremelanotide belongs to the

category of melanocortin agonists. PT-141 does not affect the vascular

system and its selective effect is limited to activation and stimulation of

melanocortin receptors to increase libido and sexual appeal.

PT-141 is a sterile, non-pyrogenic, white lyophilized powder intended for

subcutaneous or intramuscular injection, after reconstitution with sterile

Water for Injection.

Mechanism of Action

PT-141 is considered as a synthetic aphrodisiac. Alternatively to Viagra and

Cialis, it has no influence upon the vascular system, but directly increases

sexual desire. PT-141 activates the melanocortin receptors MC1R and

MC4R in the central nervous system, modulates inflammation and reduces

the restriction in blood supply to the tissues. PT-141 is a deaminated

derivative and metabolite of Melanotan II. PT-141 also acts as an agonist.

PT-141 has proved its safeness and efficiency on a broad range of patients.

Adverse reactions

PT-141 (Bremelanotide) is considered to be much safer compared to Viagra

or Cialis. However, as all other medicine it might be the reason of several

adverse reactions to occur, such as nausea, decreased appetite; flushing of

the face and increased blood pressure. The last one should not cause

discomfort for healthy individuals. Injectable PT-141 is considered not to

have this particular minor effect.

Instructions for reconstitution

Flip off the top of the peptide vial with your thumb. Use the alcohol swab to wipe the

rubber stopper of the peptide vial. Push the needle of the syringe into the middle of the

rubber stopper so it goes through the rubber and into the vial. Now, while angling the

needle so that the water for injection goes down the side of the glass, rather than

directly into the powder, inject the water for injection into the vial. Repeat this step until

you have the correct amount of water in the vial. The powder will dissolve quickly,

however it can help to gently roll the vial in between your fingers (do not shake the vial

vigorously). Remove the syringe and dispose of it. You should never reuse a syringe.

Dosage

Recommended dosage of PT-141:

• 0.30 mg (trial) — 0.70 mg (average) —  1 mg (optimal) — 1.5 mg (strong),

45 — 60 mins before sex.

Storage

• After reconstitution, may be stored for a maximum of 14 days in a refrigerator at 2°C — 8°C.
• Store vials in an upright position.
• Store in a refrigerator (2°C — 8°C). Keep in the outer carton in order to protect from light.
• For one month can be stored at room temperature.